<page_title> Pharmacology of bicalutamide </page_title> <section_title> Pharmacokinetics </section_title> <table> <cell> Css <col_header>  </col_header> </cell> <cell> 8.85 μg/mL (20.6 μmol/L) <col_header> 50 mg/day </col_header> </cell> <cell> 21.6–28.5 μg/mL (50.2–66.3 μmol/L) <col_header> 150 mg/day </col_header> </cell> </table>
At steady-state concentrations (Cₛₛ) of (R)-bicalutamide with 50 mg/day and 150 mg/day bicalutamide are 8.85 μg/mL (20.6 μmol/L) and 21.6 μg/mL (50.2 μmol/L).